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The Identification of a Sub-Micromolar Peptide-Based Protein Arginine Methyltransferase 1 (PRMT1) Inhibitor from a Plate-Based Screening Assay

  • University of North Florida

Research output: Contribution to journalArticlepeer-review

Original languageEnglish
Article number1494
JournalBiomolecules
Volume15
Issue number11
DOIs
StatePublished - Sep 23 2025

Keywords

  • Amino Acid Sequence
  • Arginine/metabolism
  • Enzyme Inhibitors/pharmacology
  • Humans
  • Kinetics
  • Methylation
  • Peptide Library
  • Peptides/chemistry
  • Protein Processing, Post-Translational
  • Protein-Arginine N-Methyltransferases/antagonists & inhibitors
  • Repressor Proteins/antagonists & inhibitors
  • Substrate Specificity

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